第1页共4页编号:时间:2021年x月x日书山有路勤为径,学海无涯苦作舟页码:第1页共4页抗肿瘤类原料药及中间体PRODUCTSPECIFICATION★原料药卡铂CarboplatinEP/USP/CP顺铂CisplatinEP/USP/CP奥沙利铂OxaliplatinEP5奈达铂NedaplatinIn-House依铂EptaplatinIn-House吉西他滨GemcitabineIn-House卡培他滨CapecitabineIn-House替加氟TegafurCP/JP吉莫斯特GimeracilIn-House氧嗪酸钾OteracilpotassiumIn-House培美曲塞二钠PemetrexedDisodiumIn-House唑来膦酸ZoledronicAcidIn-House异环膦酸铵IfosfamideUSP/CP氯法拉滨ClofarabineIn-House★中间体①铂系列药物中间体氯亚铂酸钾Potassiumtetrachloroplatinate()[10025-99-7]Ⅱ二碘二氨合铂Diiododiammineplatinum二硝基环己二胺铂DACHPLATINUMDINITRATE顺式-二氯-[反式-(-)-1,2-环己二胺]铂Cis-dichloro(trans-1-1,2-cyclohexanediamine)pt()Ⅱ左旋-反式-1,2-环己二胺(1R,2R)-(-)-1,2-diaminocyclohexane[20439-47-8]反式-1,2-环己二胺Trans-1,2-diaminocyclohexane[1121-22-8]环丁基甲酸Cyclobutanecarboxylicacid[3721-95-7]②卡培他滨中间体intermediateofCapecitabine三乙酰基-5-脱氧核糖Assay≥98.5%1,2,3-triacetyl-5-deoxy-ß-D-Ribose[62211-93-2]③吉西他滨中间体IntermediatesofGemcitabine双丙醇-D-甘露糖醇;1,2:5,6-二异亚丙基-D-mannitolAssay≥95%1,2:5,6-Bis-O-(1-methylethylidene)-D-mannitol[1707-77-3]2-脱氧-2,2-二氟戊呋喃糖-1-酮-3,5-二安息香酸盐(又名核酮糖)Assay≥95%2-Deoxy-2,2-difluoro-D-erythro-pentofuranos-1-ulose-3,5-dibenzoate[122111-01-7]第2页共4页第1页共4页编号:时间:2021年x月x日书山有路勤为径,学海无涯苦作舟页码:第2页共4页④培美曲塞二钠中间体IntermediatesofPemetrexedDisodium培美曲塞酸Pemetrexed[137281-23-3]N-(4-[2-(2-氨基-4,7-二氢-4-氧-1H-吡咯[2,3-D]嘧啶-5-基)乙基]苯甲酰)-L-谷氨酸二乙酯对甲苯磺酸盐(N-[4-[2-(2-amino-4,7-dihydro-4-oxo-3H-pyrrolo[2,3-d]pyrimidin-5-yl)ethyl]benzoyl]L-Glutamicacid[165049-28-5]4-[2-(2-氨基-4,7-二氢-4-氧-1H-吡咯[2,3-D-]嘧啶-5-基)乙基]苯甲酸4-[2-(2-amino-4-oxo-4,7-dihydro-4-oxo-3H-pyrrolo(2,3-d)pyrimidin-5-yl)ethyl]benzoicacid[137281-39-1]⑤异环磷酰胺中间体IntermediateofIfosfamide3-(2-氯乙酰基)-2-[(2-氯乙基)氨基]四氢-2H-1,3,2-恶磷-2-氧化物Ifosfamideacylationobjects[72578-71-3]⑥氯法拉滨中间体IntermediatesofClofarabine2,3,5-三苯甲酰基-ß-D-呋喃核糖beta-D-Ribofuranose2,3,5-tribenzoate[67525-66-0]1,3,5-三-O-苯甲酰基-2-脱氧-2-氟-alpha-L-阿拉伯呋喃糖1,3,5-Tri-O-benzoyl-2-deoxy-2-fluoro-alpha-L-arabinofuranosev[171721-00-9]抗真菌类原料药及中间体PRODUCTSPECIFICATION★原料药盐酸特比萘芬TerbinafineHydrochlorideEP5.3盐酸布替萘芬ButenafineHydrochlorideIn-House伏立康唑VoriconazoleIn-House★盐酸特比萘芬中间体IntermediatesofTerbinafineHydrochlorideN-甲基-1-萘甲胺N-methyl-1-naphthalenemethylamine[14489-75-9]3,3-二甲基-1-丁炔3,3-Dimethyl-1-Butyne[917-92-0]反式-1,3-二氯丙烯Trans-1,3-dichloropropene[10061-02-6]1-氯-6,6-二甲基-2-庚烯-4-炔1-chloro-6,6-dimethyl-2-heptyene-4-alkyne[126764-17-8]特比萘芬碱基Terbinafinebase抗高血压类原料药及中间体PRODUCTSPECIFICATION★原料药尼索地平NisoldipineIn-House西尼地平CilnidipineIn-House盐酸马尼地平ManidipinedihydrochlorideIn-House非洛地平FelodipineUSP30第3页共4页第2页共4页编号:时间:2021年x月x日书山有路勤为径,学海无涯苦作舟页码:第3页共4页托拉塞米TorasemideUSP30盐酸雷诺嗪RanolazinedihydrochlorideIn-House★中间体①西尼地平中间体IntermediateofCilnidipine3-氨基-2-丁烯酸肉桂酯3-AminoCrotonicAcidCinnamylEster②托拉塞米中间体IntermediateofTorasemide[4-(3-甲基苯基)氨基]吡啶-3-磺酰胺[4-(3-Methylphenyl)amino]pyridine-3-sulphonamide[72811-73-5]...