癌症靶向药(2016)肺癌靶向药疾病名称药物靶点靶向药物名称中国上市肺癌Herl(EGFR,ErbBl)Gefitinib(吉非替尼)是Erlotinib(厄洛替尼)否Osimertinib(奥斯替尼 AZD9291)Necitumumab(耐昔妥珠单Afatinib(阿法替尼)Her2(Neu,ErbB2)ALKCeritinib(赛丽替尼)Alectinib(爱乐替尼)Crizotinib(克唑替尼)是METROS1PD-1Nivolumab(纳武单抗)否Pembrolizumab(派姆单抗)VEGFR2Ramucirumab(雷莫芦单抗)VEGFBevacizumab(贝伐珠单抗)是乳腺癌靶向药疾病名称药物靶点靶向药物名称中国上市乳腺癌CDK4Palbociclib(帕博西尼)否CDK6Her2(Neu,ErbB2)Ado-trastuzumabemtansine(T-DM1)Pertuzumab(帕妥珠单抗)Trastuzumab是Herl(EGFR,ErbBl)mTORLapatiniEverolimus(曲妥珠单抗)结直肠癌靶向药疾病名称药物靶点靶向药物名称中国上市结直肠癌Her1(EGFR,ErbB1)Cetuximab(西妥西单抗)是Panitumumab(帕尼单抗)否KIT,PDGFRB,RAF,RET,
VEGFR1/2/3Regorafenib(瑞格菲尼)VEGFA/BZiv—aflibercept(阿柏西普)PIGFVEGFR2Ramucirumab(雷莫芦单抗)VEGFBevacizumab(贝伐珠单抗)是白血病靶向药疾病名称药物靶点白血病KITPDGFRABLFGFR1-3FLT3VEGFR2BTKCD20靶向药物名称中国上市Imatinib(伊马替尼)是Nilotinib(尼洛替尼)Dasatinib(达沙替尼)Bosutinib(博舒替尼)否